| Assay ID | Title | Year | Journal | Article |
|---|
| AID1271970 | Inhibition of tankyrase in human HEK293 cells assessed as decrease in non-phosphorylated beta-catenin level after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271972 | Inhibition of human TNKS2 by fluorescence analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1866927 | Inhibition of PARP1 (unknown origin) | 2022 | Journal of medicinal chemistry, 04-14, Volume: 65, Issue:7
| Small-Molecule Inhibitors of Tankyrases as Prospective Therapeutics for Cancer. |
| AID1271973 | Inhibition of tankyrase in WNT3a-stimulated human HEK293 cells by luciferase reporter gene assay | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271978 | Downregulation of TNKS1/2 expression in WNT3a-stimulated human HEK293 cells after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271971 | Inhibition of human TNKS1 by fluorescence analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271981 | Downregulation of TNKS1/2 expression in human SW480 cells after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271974 | Inhibition of tankyrase in human HEK293 cells assessed as increase in AXIN1 expression after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271975 | Downregulation of TNKS1/2 expression in human HEK293 cells after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271980 | Inhibition of tankyrase in human SW480 cells assessed as decrease in non-phosphorylated beta-catenin level after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271979 | Inhibition of tankyrase in human SW480 cells assessed as increase in AXIN1 expression after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1271976 | Inhibition of tankyrase in WNT3a-stimulated human HEK293 cells assessed as increase in AXIN1 expression after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1866926 | Inhibition of TNKS2 (unknown origin) | 2022 | Journal of medicinal chemistry, 04-14, Volume: 65, Issue:7
| Small-Molecule Inhibitors of Tankyrases as Prospective Therapeutics for Cancer. |
| AID1271977 | Inhibition of tankyrase in WNT3a-stimulated human HEK293 cells assessed as decrease in non-phosphorylated beta-catenin level after 24 hrs by western blot analysis | 2016 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 26, Issue:2
| Development and structural analysis of adenosine site binding tankyrase inhibitors. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID588519 | A screen for compounds that inhibit viral RNA polymerase binding and polymerization activities | 2011 | Antiviral research, Sep, Volume: 91, Issue:3
| High-throughput screening identification of poliovirus RNA-dependent RNA polymerase inhibitors. |
| AID540299 | A screen for compounds that inhibit the MenB enzyme of Mycobacterium tuberculosis | 2010 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 20, Issue:21
| Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | 2014 | Journal of biomolecular screening, Jul, Volume: 19, Issue:6
| A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum. |
| AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | | | |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |